Medical Attributes of Serenoa repens - Saw palmetto

By Christa Filipkowski, Barbara DiCaprio, and Brielle Stanton
Wilkes University, Wilkes-Barre, PA

July, 2011

Serenoa repens is a small shrub belonging to the palm family Arecaceae.  Commonly known as the saw palmetto or American dwarf palm, it is found in low pinewoods, savannas, and thickets in the southeastern US, from South Carolina to Florida, and west to Mississippi.  S. repens has above-ground horizontal stems, palmately compound green leaves that bear saw-like teeth on the petiole, white flowers that bloom in late spring, and black drupes that each hold a single seed (Foster & Duke 2000).


Native Americans once regularly consumed S. repens fruit (Foster & Duke 2000) and used it to treat genitourinary disorders, mucous membrane inflammation, testosterone deficiency in males, or to increase breast size in females (Suzuki et al. 2009).  Extracts were also traditionally used to relieve colds, coughs, asthma, migraines, and chronic bronchitis (Foster & Duke 2000).


Today, S. repens is still used to remedy genitourinary disorders, to increase sperm production or breast size, as an aphrodisiac, and as a mild diuretic (Suzuki et al. 2009).  Specifically, extracts of S. repens’ fruits are most often administered to treat benign prostatic hyperplasia (BPH) and associated lower urinary tract symptoms (LUTS), which are conditions that are frequent in aging men (Suzuki et al. 2009, Ernst 2002, Lee et al. 2009).  BPH is enlargement of the prostate gland, which can cause obstructions in the lower urinary tract, making it difficult to urinate (Tacklind et al. 2009). 


S. repens contains multiple chemical compounds that have been useful in BPH therapy management.  For instance, the berry lipid extract (BLE) has shown increasing promise in the inhibition of the enzyme 5-alpha-reductase (Angwafor 2008), which blocks the conversion of testosterone to dihydrotesterone and can thereby reduce BPH (Wargo et al. 2010).  The specific active constituents within the berry lipid extract include sterols and free fatty acids (Gordon & Shanughnessy 2003).


A study comparing in vitro and in vivo analysis of this therapeutic plant proved that the combination of S. repens, lycopene and selenium could be effective in BPH treatments as it increases the anti-inflammatory nature of S. repens compounds (Bonvissuto et al. 2011).  Randomized clinical trials on male BPH sufferers have proven that an herbal blend of the plant can be a safe and successful treatment for moderately symptomatic cases of BPH (Marks et al. 2000, Hong et al. 2009).  The combination of anti-androgenic, anti-inflammatory, and anti-edema effects has shown useful in therapy management (Suzuki et al. 2009).   S. repens has been examined as a form of phytotherapy for other prostate disorders, including prostate cancer, as it may be useful in inhibiting the production of new tumors (tumorigenesis) (Sosnowska & Balslev 2009).


S. repens extract has also been proven to increase sexual function (Sinescu et al. 2011), to reduce both intra- and postoperative complications in BPH surgeries, including transurethral resection of the prostate and open prostatectomy (Anceschi et al. 2010), and to treat chronic pelvic pain syndrome (Morgia et al. 2010).


Aside from their application to disorders of the urogenital system, liposterolic extract from the saw palmetto combined with two anti-inflammatory agents, carnitine and thiocitic acid, effectively controlled chronic inflammation of hair follicles in cases of androgenetic aplopecia (AGA), or male pattern balding.  Beta-sitosterol was the specific S. repens compound studied, and had demonstrated in in vitro simulations of human keratinocytes (Chittur et al. 2009). 


The adverse events associated with the use of S. repens are mild and similar to those expected with the placebo.  The most frequently reported adverse events are abdominal pain, diarrhea, nausea, fatigue, headache, decreased libido and rhinitis (Agbabiaka et al. 2009). No drug interactions have been reported with S. repens, which makes it a suitable therapy candidate (Izzo & Ernst 2009, Gordon & Shanughnessy 2003).  However, if used as a form of self-medication, there is a risk of missing the early detection of prostate cancer (Murugusundram 2009).


Serenoa repens has been used as a safe treatment option for benign prostate hyperplasia and associated lower urinary tract sypmtoms, as well as androgenetic aplopecia.  S. repens is tolerated by most users and is not associated with any serious side effects.  As with all botanical therapies, a physician should be made aware of S. repens supplements and can determine a correct dosage for an individual patient.

LITERATURE CITED

Agbabiaka, T.B., M.H. Pittler, B. Wider, et al. 2009. Serenoa repens (saw palmetto): a systematic review of adverse events. Drug Saf. 32(8):637-47

 

Anceschi, R., M. Bisi, N. Ghidini, et al. 2010. Serenoa repens (Permixon) reduces intra- and postoperative complications of surgical treatments of benign prostatic hyperplasia. Minerva Urol Nefrol. 62(3):219-23.

 

Angawafor, F., & M.L. Anderson. 2008. An open label, dose response study to determine the effect of a dietary supplement on dihydrotestosterone testosterone, and estradiol levels in healthy males. J Int Soc Sports Nutrition 12:5:12.

 

Bonvissuto, G., L. Minutoli, G. Morgia, et al. 2011. Effect of Serenoa repens, lycopene, and selenium on proinflammatory phenotype activation: an in vitro and in vivo comparison study. Urology 77(1):248.e9-16.

 

Chittur, S., B. Parr, & G. Marcovici. 2009. Inhibition of inflammatory gene expression in keratinocytes using a composition containing carnitine, thioctic acid and saw palmetto extract.  Evidence Based Complementary Alternative Medicine. Epub ahead of print.

 

Ernst, E.  2002. The risk-benefit profile of commonly used herbal therapies: Ginkgo, St. John’s Wort, Ginseng, Echinacea, Saw Palmetto, and Kava.  Ann Internal Medicine 1:136(1):42-53.           

 

Foster, S., & J.A. Duke.  2000. Eastern/Central Medicinal Plants and Herbs. Houghton Mifflin Co. New York. 411 pp.

 

Gordon, A.E., & A. F. Shanughnessy. 2003. Saw palmetto for prostate disorders. American Family Physician 15:67(6):1281-3.

 

Hong, H., C. Kim, & S. Maeng. 2009. Effects of pumpkin seed oil and saw palmetto oil in Korean men with symptomatic benign prostatic hyperplasia. Nutr Res Pract 3:323-327.

 

Izzo, A.A. & E. Ernst.  2009. Interactions between herbal medicines and prescribed drugs: an updated systematic review. Drugs 13:1777-98.

 

Lee, J., G. Andriole, A. Avins, et al. 2009. Redesigning a large-scale clinical trial in response to negative external trial results:  the CAMUS study of phytotherapy for benign prostatic hyperplasia.  Clin Trials. 6(6):628-36.

 

Marks, L.S., A. W. Partin, J.I. Epstein, et al. 2000. Effects of a saw palmetto herbal blend in men with symptomatic benign prostatic hyperplasia. J Urol. 163(5):1451-6.

 

Morgia, G., G. Mucciardi, A. Gali, et al. 2010. Treatment of chronic prostatitis/chronic pelvic pain syndrome category IIIA with Serenoa repens plus selenium and lycopene (Profluss) versus S. repens alone: an Italian randomized multicenter-controlled study. Urol Int. 84(4):400-6.

 

Murugusundram, S.  2009. Serenoa repens: Does it have any role in the management of androgenetic alopecia?  J Cutan Aesthet Surg. 2(1):31-2.

 

Sinescu, I., P. Geavlete, R. Multescu, et al. 2011. Long-term efficacy of Serenoa repens treatment in patients with mild and moderate symptomatic benign prostatic hyperplasia. Urol Int. 86(3):284-9.

 

Sosnowska, J., & H. Balslev. 2009. American palm ethnomedicine: a meta-analysis.  J Ethnobiol Ethnomedicine 24:5;43

 

Suzuki, M., Y. Ito, T. Fujino, et al. 2009. Pharmacological effects of saw palmetto extract in the lower urinary tract. Acta Pharmacol Sin. 30(3):227-81.

 

Tacklind, J., R. MacDonald, I. Rutks, et al. 2009. Serenoa repens for benign prostatic hyperplasia.  Cochrane Database Syst Rev. 15:(2):CD001423.

 

Wargo, K.A., E. Allman, F. Ibrahim. 2010. A possible case of saw palmetto-induced pancreatitis. South Med J. 103(7):683-5.

 

Yang, Y., T. Ikezoe, Z. Zheng, et al. 2007. Saw palmetto induces growth arrest and apoptosis of androgen-dependent prostate cancer LNCaP cells via inactiviation of STAT 3 and androgen receptor signaling. Int J Oncol. 31(3):593-600.


This paper was developed as part of the BIO 368 - Medical Botany course offered at Wilkes University during the summer of 1999. Course instructor was Kenneth M. Klemow, Ph.D. (kklemow@wilkes.edu). The information contained herein is based on published sources, and is made available for academic purposes only. No warrantees, expressed or implied, are made about the medical usefulness or dangers associated with the plant species in question.

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This page posted and maintained by Kenneth M. Klemow, Ph.D., Biology Department, Wilkes University, Wilkes-Barre, PA 18766. (570) 408-4758, kklemow@wilkes.edu.